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Synthesis of Quinazolin-4(3H)-Ones Via the Reaction of Isatoic Anhydride With Benzyl Azides in the Presence of Potassium Tert-Butoxide in Dmso Publisher



Sayahi MH1 ; Bahadorikhalili S2 ; Mahdavi M3 ; Baghshirin L1
Authors

Source: Chemistry of Heterocyclic Compounds Published:2019


Abstract

[Figure not available: see fulltext.] In this paper, a novel method is described for the synthesis of quinazolin-4(3H)-one derivatives via the reaction of isatoic anhydride with benzyl azides in the presence of potassium tert-butoxide in DMSO. The reaction is completed after 4 h at 100°C to produce the title products in good yields. © 2019, Springer Science+Business Media, LLC, part of Springer Nature.
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