A Novel and Efficient Synthesis of 2-Substituted Quinazolin-4(3H)-Ones by the Reaction of (Het)Arylmethanamines With Isatoic Anhydride

A Novel and Efficient Synthesis of 2-Substituted Quinazolin-4(3H)-Ones by the Reaction of (Het)Arylmethanamines With Isatoic Anhydride Publisher

Mahdavi M¹ ; Hassanzadeh R² ; Soheilizad M² ; Golshani S² ; Moghimi S² ; Firoozpour L¹ ; Shafiee A² ; Foroumadi A^{1, 2}

Source: Tetrahedron Letters Published:2016

Abstract

A novel and straightforward method for the synthesis of quinazolin-4(3H)-ones is described. The one-pot reaction between isatoic anhydride and (het)arylmethanamines led to the formation of N-substituted anthranilamides, which under aerobic conditions in the presence of CuBr undergo an in situ oxidation–cyclization reaction to produce quinazolin-4(3H)-ones in good yields. © 2016 Elsevier Ltd

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Mohammad Mahdavi (17)

Alireza Foroumadi (6)

Style	Citing Format
MLA	Mahdavi M, et al.. "A Novel and Efficient Synthesis of 2-Substituted Quinazolin-4(3H)-Ones by the Reaction of (Het)Arylmethanamines With Isatoic Anhydride." Tetrahedron Letters, vol. 57, no. 33, 2016, pp. 3770-3772.
APA	Mahdavi M, Hassanzadeh R, Soheilizad M, Golshani S, Moghimi S, Firoozpour L, Shafiee A, Foroumadi A (2016). A Novel and Efficient Synthesis of 2-Substituted Quinazolin-4(3H)-Ones by the Reaction of (Het)Arylmethanamines With Isatoic Anhydride. Tetrahedron Letters, 57(33), 3770-3772.
Chicago	Mahdavi M, Hassanzadeh R, Soheilizad M, Golshani S, Moghimi S, Firoozpour L, Shafiee A, Foroumadi A. "A Novel and Efficient Synthesis of 2-Substituted Quinazolin-4(3H)-Ones by the Reaction of (Het)Arylmethanamines With Isatoic Anhydride." Tetrahedron Letters 57, no. 33 (2016): 3770-3772.
Harvard	Mahdavi M et al. (2016) 'A Novel and Efficient Synthesis of 2-Substituted Quinazolin-4(3H)-Ones by the Reaction of (Het)Arylmethanamines With Isatoic Anhydride', Tetrahedron Letters, 57(33), pp. 3770-3772.
Vancouver	Mahdavi M, Hassanzadeh R, Soheilizad M, Golshani S, Moghimi S, Firoozpour L, et al.. A Novel and Efficient Synthesis of 2-Substituted Quinazolin-4(3H)-Ones by the Reaction of (Het)Arylmethanamines With Isatoic Anhydride. Tetrahedron Letters. 2016;57(33):3770-3772.
BibTex	@article{ author = {Mahdavi M and Hassanzadeh R and Soheilizad M and Golshani S and Moghimi S and Firoozpour L and Shafiee A and Foroumadi A}, title = {A Novel and Efficient Synthesis of 2-Substituted Quinazolin-4(3H)-Ones by the Reaction of (Het)Arylmethanamines With Isatoic Anhydride}, journal = {Tetrahedron Letters}, volume = {57}, number = {33}, pages = {3770-3772}, year = {2016} }
RIS	TY - JOUR AU - Mahdavi M AU - Hassanzadeh R AU - Soheilizad M AU - Golshani S AU - Moghimi S AU - Firoozpour L AU - Shafiee A AU - Foroumadi A TI - A Novel and Efficient Synthesis of 2-Substituted Quinazolin-4(3H)-Ones by the Reaction of (Het)Arylmethanamines With Isatoic Anhydride JO - Tetrahedron Letters VL - 57 IS - 33 SP - 3770 EP - 3772 PY - 2016 ER -

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